L-803087

Term ID

CHEBI:177197

Synonyms

L 803087
L-803,087
L803087
methyl (2S)-5-carbamimidamido-2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanamido]pentanoate
methyl N(2)-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanoyl]-L-argininate
N(2)-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginine methyl ester

Definition

A fluoroindole that is 1H-indole substituted by phenyl, 4-{[(2S)-5-carbamimidamido-1-methoxy-1-oxopentan-2-yl]amino}-4-oxobutyl, fluoro and fluoro groups at positions 2, 3, 5 and 7, respectively. It is a selective nonpeptidic agonist of the somatostatin subtype-4 (SST4) receptor with Ki of 0.7 nM.

References

Ontology

ChEBI ( EBI )

Relationships

is a type of: benzenes fluoroindole guanidines L-arginine derivative methyl ester ... Show All 7 Terms

benzenes fluoroindole guanidines L-arginine derivative methyl ester phenylindole secondary carboxamide Show first 5 Terms
has_role: somatostatin receptor agonist

somatostatin receptor agonist Show first 5 Terms

Phenotype

Phenotype resulting from L-803087

Phenotype where environments contain L-803087

Phenotype modified by environments containing L-803087

Human Disease Model