PUBLICATION

Stereocontrol of arachidonic acid oxygenation by vertebrate lipoxygenases, newly cloned zebrafish lipoxygenase1 does not follow the A-vs-G concept

Authors
Jansen, C., Hofheinz, K., Vogel, R., Anton, M., Reddanna, P., Kuhn, H., and Walther, M.
ID
ZDB-PUB-110907-9
Date
2011
Source
The Journal of biological chemistry   286(43): 37804-12 (Journal)
Registered Authors
Keywords
eicosanoid, enzyme catalysis, leukotriene, lipid oxidation, lipoxygenase pathway, zebrafish, enantioselectivity, stereochemistry
MeSH Terms
  • Animals
  • Arachidonic Acid/genetics
  • Arachidonic Acid/metabolism*
  • Humans
  • Isoenzymes/genetics
  • Isoenzymes/metabolism
  • Lipoxygenase/genetics
  • Lipoxygenase/metabolism*
  • Macaca mulatta
  • Mice
  • Pongo
  • Rabbits
  • Species Specificity
  • Zebrafish/genetics
  • Zebrafish/metabolism*
  • Zebrafish Proteins/genetics
  • Zebrafish Proteins/metabolism*
PubMed
21880725 Full text @ J. Biol. Chem.
Abstract
Animal lipoxygenases (LOX) are classified according to their specificity of arachidonic acid oxygenation and previous sequence alignments suggested that S-LOX contain a conserved Ala at a critical position at the active site but R-LOX carry a Gly instead. Here we cloned, expressed and characterized a novel LOX-isoform from the model vertebrate Danio rerio (zebrafish) that carries a Gly at this critical position classifying this enzyme as putative arachidonic acid R-LOX. Surprisingly, the almost exclusive arachidonic acid oxygenation product was 12S-H(p)ETE and extensive mutation around G410 failed to induce R-lipoxygenation. This finding prompted us to explore the importance of the corresponding amino acids in other vertebrate S-LOXs. We found that A-to-G exchange in human 15-LOX2 and human platelet 12-LOX induced major alterations in the reaction specificity with an increase of specific R-oxygenation products. For mouse 5-LOX, for 12/15-LOX from rabbits, men, rhesus monkeys, orang-utans and mice only minor alterations in the reaction specificity were observed. For these enzymes S-HETE isomers remained the major oxygenation products whereas chiral R-HETEs contributed only 10-30% to the total product mixture. Taken together this data indicates that the A-vs-G concept may not always predict the reaction specificity of vertebrate LOX-isoforms.
Genes / Markers
Figures
Expression
Phenotype
Mutations / Transgenics
Human Disease / Model
Sequence Targeting Reagents
Fish
Antibodies
Orthology
Engineered Foreign Genes
Mapping